ホーム 計算ツール
代理店ログイン
製品 阻害剤 ライブラリー リコンビナントタンパク質 キット サービス お問い合わせ
ペプチド 抗体 色素試薬 PROTAC バーチャルスクリーニング TargetMolキット Cell Counting Kit-8 (CCK-8) Inhibitor Cocktails 天然化合物 フェノール類 アルカロイド類 フラボノイド類
阻害剤 血管新生 アポトーシス オートファジー 細胞周期・チェックポイント クロマチン・エピジェネティック 細胞骨格シグナル DNA損傷・DNA修復 内分泌・ホルモン GPCR/Gタンパク質 免疫・炎症 JAK・STATシグナル MAPK
膜輸送体・イオンチャネル 代謝 微生物学・ウィルス学 神経科学 NF-Κb 酸化還元 PI3K/Akt/mTORシグナル プロテアーゼ・プロテアソーム 幹細胞 チロシンキナーゼ・アダプター ユビキチン PROTAC
化合物ライブラリー 生物活性化合物ライブラリー ゼネラルバイオウアクティヴライブラリー 承認/再開発 医薬品ライブラリー 疾患別 化合物ライブラリー 標的/経路別 化合物ライブラリー 特徴的な生物活性化合物ライブラリー 天然化合物ライブラリー HTS用天然物ライブラリー 分野別 天然化合物ライブラリー 天然物誘導体ライブラリー CADD用天然物ライブラリー ドラッグライク 化合物ライブラリー フラグメントライブラリー カスタム化合物ライブラリー
シグナル伝達経路 血管新生 アポトーシス オートファジー 細胞周期・チェックポイント クロマチン・エピジェネティック 細胞骨格シグナル
DNA損傷・DNA修復 内分泌・ホルモン GPCR/Gタンパク質 免疫・炎症 JAK・STATシグナル MAPK 膜輸送体・イオンチャネル
代謝 微生物学・ウィルス学 神経科学 NF-Κb 酸化還元 PI3K/Akt/mTORシグナル プロテアーゼ・プロテアソーム
幹細胞 チロシンキナーゼ・アダプター ユビキチン その他 PROTAC
生物活性化合物ライブラリー ゼネラルバイオウアクティヴライブラリー 承認/再開発 医薬品ライブラリー 疾患別 化合物ライブラリー 標的/経路別 化合物ライブラリー 特徴的な生物活性化合物ライブラリー
天然化合物ライブラリー HTS用天然物ライブラリー 分野別 天然化合物ライブラリー 天然物誘導体ライブラリー CADD用天然物ライブラリー
ドラッグライク 化合物ライブラリー ドラッグライクライブラリー
フラグメントライブラリー ゼネラルフラグメントライブラリー 特徴的なフラグメントライブラリー カスタム化合物ライブラリー
Cytokines and Growth Factors •   Cytokines •   Growth Factors Receptor Proteins •   Fc Receptors •   Cytokines and Growth Factor Receptors
CD Proteins •   T Cell CD Proteins •   B Cell CD Proteins Immune Checkpoint Proteins •   Co-inhibitory Immune Checkpoint Proteins •   Co-stimulatory Immune Checkpoint Proteins
CAR-T Therapy Target Proteins •   Hematologic Malignancies Target Proteins •   Solid Tumors Target Proteins Enzymes •   Oxidoreductases,EC 1 •   Transferases,EC 2
Viral Proteins •   Coronavirus (CoV) Proteins •   Influenza Proteins Fluorescent Proteins Others

検索結果

Search Results for " Fatty Acid Synthase (FASN) "

ターゲット

Fatty Acid Synthase

23

阻害剤

9

天然化合物

1

ライブラリー

カタログ番号 製品名 別名 ターゲット
T11557 FASN-IN-3 Fatty Acid Synthase
FASN-IN-3 is an inhibitor of fatty acid synthase (FASN).
T11267 FASN-IN-1 TVB-2460 Fatty Acid Synthase
FASN-in-1 is an effective, specific inhibitor of fatty acid synthase (FASN), a compound specifically designed to target and inhibit the activity of the enzyme involved in fatty acid synthesis, potentially disrupting fatt...
T7947 FT113 Fatty Acid Synthase
FT113 is a novel potent inhibitor of fatty acid synthase (fasn, IC50 : 213 nM),and exhibits anti-cancer activity
T0686 Orlistat Ro-18-0647,Tetrahydrolipstatin Apoptosis , Others , Fatty Acid Synthase
Orlistat (Tetrahydrolipstatin) is an Intestinal Lipase Inhibitor. The mechanism of action of orlistat is as a Lipase Inhibitor.
T17181 TVB-3664 Fatty Acid Synthase
TVB-3664 significantly decreases tubulin palmitoylation and mRNA expression. TVB-3664 is a reversible and highly bioavailable fatty acid synthase inhibitor (IC50: 18 nM and 12 nM for human and mouse cell palmitate synthe...
T17180 TVB-3166 Apoptosis , Others , Fatty Acid Synthase
TVB-3166 induces apoptosis and inhibits in-vivo xenograft tumor growth. TVB-3166 is a reversible and selective fatty acid synthase inhibitor (IC50s: 42 nM and 81 nM for biochemical FASN and cellular palmitate synthesis,...
T7798 FGH10019 FGH-10019 NPC1L1 , Fatty Acid Synthase
FGH10019 is a novel inhibitor of sterol regulatory element-binding protein (SREBP) ( IC50 :1 μM).
T15271 Denifanstat FASN-IN-2,TVB2640,TVB-2640 Fatty Acid Synthase
Denifanstat (FASN-IN-2) is a Fatty Acid Synthase (FASN) inhibitor(IC50 of 0.052 μM and an EC50 of 0.072 μM),with potential antineoplastic activity.
T9266 Fatostatin Lipid , Fatty Acid Synthase
Fatostatin is a specific inhibitor of SREBP activation, it impairs the activation of SREBP-1 and SREBP-2. Fatostatin binds to SCAP (SREBP cleavage-activating protein), and inhibits the ER-Golgi translocation of SREBPs.
T12437 PF429242 dihydrochloride S1P Receptor
PF429242 dihydrochloride is a reversible and competitive inhibitor of S1P (IC50 of 175 nM).
T36841 IPI-9119 Fatty Acid Synthase
IPI-9119 is an orally active, selective and irreversible FASN inhibitor (IC50 = 0.3 nM).
T10656 Trans-C75 (±)-C75 Others , Fatty Acid Synthase
trans-C75 ((±)-C75) is an enantiomer of C75. C75 is an inhibitor of fatty-acid synthase (FASN).
T6832 Fatostatin hydrobromide Fatostatin HBr,Fatostatin A,Fatostatin A HBr,Fatostatin NPC1L1 , Fatty Acid Synthase
Fatostatin hydrobromide (Fatostatin A HBr) ia an inhibitor of sterol regulatory element binding protein (SREBP). It impairs the activation of SREBP-1 and SREBP-2.
T10657 C75 C-75 Fatty Acid Synthase
C75 is an inhibitor synthetic fatty-acid synthase (FASN) and inhibits prostate cancer cells PC3 (IC50: 35 μM).
T15429 GSK2194069 Others , NADPH , Fatty Acid Synthase
GSK2194069 is an active β-keto reductase (KR)-specific inhibitor of fatty acid synthase (FASN) with an IC50 of 7.7 nM in an assay for the detection of released CoA.GSK2194069 inhibits the proliferation of FAS in cancer c...
T21831 UCM05 G28UCM Fatty Acid Synthase
UCM05 (G28UCM) is a potent inhibitor of fatty acid synthase (FASN) with efficacy against HER2+ breast cancer xenografts, including in cell lines resistant to anti-HER2 drugs [1]. Additionally, it functions as an inhibito...
T11574 HS79 Others
T11575 HS80 Others
T37776 FASN-IN-4 tosylate
FASN-IN-4 tosylate is a potent fatty acid synthase (FASN) inhibitor, exhibiting an IC50 value of 10 nM. Additionally, it demonstrates inhibitory activity against SARS-CoV-2, with an EC50 of 18.6 nM [2].
T70978 5-Hydroxy Lansoprazole Sulfide
5-Hydroxy Lansoprazole Sulfide is an inhibitor of fatty acid synthase (FASN). FASN, which is responsible for de-novo synthesis of lipids, has been found to be overexpressed in cancerous tissue. 5-Hydroxy Lansoprazole Sul...
T78872 CTL-06
CTL-06, a Fatty Acid Synthase (FASN) inhibitor with an IC50 of 3 μM, induces apoptosis, while CTL-12 impedes cell cycle progression in the Sub-G1/S phase and modulates apoptotic and anti-apoptotic markers by upregulating...
T78873 CTL-12
CTL-12, a fatty acid synthase (FASN) inhibitor (IC50: 2.5 μM), induces apoptosis and disrupts the cell cycle at the Sub-G1/S phase. It upregulates caspase-9 and the apoptosis marker Bax, while downregulating the anti-apo...
T70882 Orlistat-d3
Orlistat-d3 is intended for use as an internal standard for the quantification of orlistat by GC- or LC-MS. Orlistat is a digestive lipase inhibitor. It inhibits diacylglycerol lipase α (DAGLα), DAGLβ, α/β-hydrolase doma...
カタログ番号 製品名 別名 ターゲット
TQ0260 Cerulenin Antibiotic , Antifungal , Fatty Acid Synthase
Cerulenin is a natural inhibitor of fatty acid synthase (FAS). It is produced by the fungus Cephalosporium caeruleus.
T2824 Pedunculoside Others , Fatty Acid Synthase
Pedunculoside is extracted from Ilex rotunda Thunb.
T5S0246 Pseudoprotodioscin Others , Fatty Acid Synthase
1. Pseudoprotodioscin has moderate cytotoxicity.
TJS0387 Desoxyrhaponticin Deoxyrhapontin,Deoxyrhaponticin Apoptosis , Fatty Acid Synthase
1. Desoxyrhaponticin (Deoxyrhaponticin) is an agent that is potentially effective in controlling postprandial hyperglycemia in diabetes, the in vivo antidiabetic action of this compound can be explained, in part at least...
T3121 Betulin Trochol,betulinic alcohol,betuline,betulinol,Betulol Apoptosis , Endogenous Metabolite , Lipid , Fatty Acid Synthase
Betulin (betulinol) (lup-20(29)-ene-3β, 28-diol) is an abundant, naturally occurring triterpene. It is commonly isolated from the bark of birch trees where it forms up to 30% of the dry weight of the extractive and is fo...
T3322 Trans-Chalcone Chalcone,Cinnamophenone,Chalkone Apoptosis , Others , Antifungal , Fatty Acid Synthase
trans-Chalcone (Chalkone) is an aromatic ketone that forms the central core for a variety of important biological compounds, which are known collectively as chalcones.
T3324 Lycorine Galanthidine,Narcissine,Amarylline,Belamarine,Licorine Apoptosis , Virus Protease , Antibacterial , AChR , Fatty Acid Synthase
Lycorine (Narcissine) inhibits protein synthesis and may inhibit ascorbic acid biosynthesis, although studies on the latter are controversial and inconclusive.
T4S1173 Agrimol B Sirtuin , PPAR
1. Agrimol B is a main active ingredient isolated from Agrimonia pilosa Ledeb.
T4S1421 Praeruptorin B Praeruptorin D NPC1L1 , Fatty Acid Synthase
Praeruptorin B is an inhibitor of sterol regulatory element-binding proteins (SREBPs). It can also significantly up-regulate CYP3A4 expression and activity via the PXR-mediated pathway.

天然物製品

Cerulenin
TQ0260
Synonym:
Target: Antibiotic, Antifungal, Fatty Acid Synthase
Pedunculoside
T2824
Synonym:
Target: Others, Fatty Acid Synthase
Pseudoprotodioscin
T5S0246
Synonym:
Target: Others, Fatty Acid Synthase
Desoxyrhaponticin
TJS0387
Synonym: Deoxyrhapontin,Deoxyrhaponticin
Target: Apoptosis, Fatty Acid Synthase
Betulin
T3121
Synonym: Trochol,betulinic alcohol,betuline,betulinol,Betulol
Target: Apoptosis, Endogenous Metabolite, Lipid, Fatty Acid Synthase
trans-Chalcone
T3322
Synonym: Chalcone,Cinnamophenone,Chalkone
Target: Apoptosis, Others, Antifungal, Fatty Acid Synthase
Lycorine
T3324
Synonym: Galanthidine,Narcissine,Amarylline,Belamarine,Licorine
Target: Apoptosis, Virus Protease, Antibacterial, AChR, Fatty Acid Synthase
Agrimol B
T4S1173
Synonym:
Target: Sirtuin, PPAR
Praeruptorin B
T4S1421
Synonym: Praeruptorin D
Target: NPC1L1, Fatty Acid Synthase
カタログ番号 製品名
L2510 Lipid Metabolism Compound Library

496 compounds
A unique collection of 496 compounds targeting lipid metabolism, can be used for high-throughput screening (HTS) and high-content screening (HCS).

ライブラリー

Lipid Metabolism Compound Library
L2510
Compounds: 496
TARGETMOLについて
会社情報 プライバシー保護について イベント＆ニュース 利用規約
サポート
お問い合わせ 代理店情報 品質管理 技術サポート
技術資料
製品カタログ 引用文献 シグナル伝達経路 溶解計算
ニュースレター登録
ニュースレターで最新の製品情報やお得な情報をお届けします。
ニュースレターで最新の製品情報やお得な情報をお届けします。
TargetMolについて
サポート
技術資料
本ウェブサイトに掲載されている製品は全て研究用試薬です。研究目的以外の用途にはご使用できません。
Copyright © 2015-2023 TargetMol Chemicals Inc. All rights reserved.